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The paper by Hosono-san, Kamakura-san, and Tanifuji on the scaffold redesign of Ecteinascidin 743 has been published in Chem! This work was conducted in collaboration with research groups led by Prof. Sota Sato (UTokyo), Dr. Hiroyuki Seimiya, and Dr. Shingo Dan (Japanese Foundation For Cancer Research).

Tanifuji, R.*; Hosono, E.; Kamakura, H.; Muramatsu, Y.; Yoshida, S.; Sato, S.; Ohashi, Y.; Dan, S.; Seimiya, H.*; Oguri, H.*

Strategic Scaffold Redesign of Ecteinascidins: An Approach for Generating Anticancer Macrocycles.

DOI: 10.1016/j.chempr.2025.102664


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Nikkei web 日本経済新聞 web: 東大、がん研究会と共同で抗がん剤エクテナサイジンの骨格を再設計しマクロ環状中分子群を短工程で創製する合成プロセスを開発

(2025.07.19)